| AZD0837 | AstraZeneca | Phase 1 | Completed | |
| Valsartan | Novartis | Phase 1 | Completed | |
| ALT02 + EU-licensed Herceptin + US-licensed Herceptin | Alteogen | Phase 1 | Completed | |
| Lasmiditan + Placebo | Eli Lilly | Phase 1 | Completed | |
| LOXO-783 | Eli Lilly | Phase 1 | Completed | |
| LY2541546 - IV + LY2541546 - SC + Placebo | Eli Lilly | Phase 1 | Completed | |
| LY3867070 + Placebo | Eli Lilly | Phase 1 | Recruiting | |
| Mirikizumab Test + Mirikizumab Test + Mirikizumab Reference | Eli Lilly | Phase 1 | Completed | |
| [¹⁴C]-LY3484356 + LY3484356 + [¹⁴C]-LY3484356 (IV) | Eli Lilly | Phase 1 | Completed | |
| Ixekizumab | Eli Lilly | Phase 1 | Completed | |
| Lasmiditan + Propranolol | Eli Lilly | Phase 1 | Completed | |
| LY3537982 + Digoxin + Rosuvastatin + Midazolam + Midazolam | Eli Lilly | Phase 1 | Completed | |
| LY3074828 | Eli Lilly | Phase 1 | Completed | |
| [(11)C] MePPEP | Eli Lilly | Phase 1 | Completed | |
| LY3451838 + LY3451838 + LY3451838 + LY3451838 + LY3451838 + LY3451838 + LY3451838 + Placebo | Eli Lilly | Phase 1 | Completed | |
| LY3537031 | Eli Lilly | Phase 1 | Recruiting | |
| LY2963016 | Eli Lilly | Phase 1 | Completed | |
| Baricitinib suspension + Baricitinib tablet | Eli Lilly | Phase 1 | Completed | |
| [14C]-LY3866288 + LY3866288 + [14C]-LY3866288 | Eli Lilly | Phase 1 | Completed | |
| Selpercatinib + Moxifloxacin + Placebo | Eli Lilly | Phase 1 | Completed | |
| LY3502970 + Esomeprazole | Eli Lilly | Phase 1 | Completed | |
| LY3375880 IV + LY3375880 SC + Placebo IV + Placebo SC | Eli Lilly | Phase 1 | Completed | |
| Midazolam + Selpercatinib | Eli Lilly | Phase 1 | Completed | |
| LY3214996 + [14C]-LY3214996 | Eli Lilly | Phase 1 | Completed | |
| LY3871801 + Placebo | Eli Lilly | Phase 1 | Completed | |
| LY3305677 + Placebo | Eli Lilly | Phase 1 | Completed | |
| Selpercatinib | Eli Lilly | Phase 1 | Completed | |
| LY3209590 (SC) + LY3209590 (IV) | Eli Lilly | Phase 1 | Completed | |
| LY3819253 + Placebo | Eli Lilly | Phase 1 | Completed | |
| [14C]-LY3556050 | Eli Lilly | Phase 1 | Completed | |
| LY3540378 + Placebo + LY3540378 | Eli Lilly | Phase 1 | Completed | |
| Orforglipron + Midazolam + Quinidine | Eli Lilly | Phase 1 | Completed | |
| Mirikizumab | Eli Lilly | Phase 1 | Recruiting | |
| LY3437943 | Eli Lilly | Phase 1 | Completed | |
| LY4086940 + Placebo + LY4086940 | Eli Lilly | Phase 1 | Recruiting | |
| Pegilodecakin | Eli Lilly | Phase 1 | Completed | |
| Rosuvastatin + Selpercatinib | Eli Lilly | Phase 1 | Completed | |
| LY4100511 | Eli Lilly | Phase 1 | Completed | |
| V930 | Merck | Phase 1 | Completed | |
| E2609 + Placebo | Eisai | Phase 1 | Completed | |
| LY3971297 + Placebo + LY3971297 IV | Eli Lilly | Phase 1 | Recruiting | |
| Selpercatinib + Omeprazole | Eli Lilly | Phase 1 | Completed | |
| LY3471851 | Eli Lilly | Phase 1 | Completed | |
| LY3372689 | Eli Lilly | Phase 1 | Completed | |
| Lebrikizumab + Placebo | Eli Lilly | Phase 1 | Completed | |
| LY4065967 | Eli Lilly | Phase 1 | Completed | |
| CTL02 + CTL0201 + CTL0202 | Celltrion | Phase 1 | Completed | |
| CT-L01 12.5/1,000 mg + CT-L01 12.5/1,000 mg | Celltrion | Phase 1 | Completed | |
| CT-P6 SC + EU-Approved Herceptin SC | Celltrion | Phase 1 | Active | |
| L04RD1 + L04TD1 + L04TD1 + L04RD1 | Celltrion | Phase 1 | Completed | |
| CT-G11 + CT-G20 + CT-G11 Placebo + CT-G20 Placebo | Celltrion | Phase 1 | Completed | |
| CT-P17 + US-licensed Humira + EU-approved Humira | Celltrion | Phase 1 | Completed | |
| CT-L01 + Alogliptin Benzoate 25 mg + Metformin HCl XR 1,000 mg | Celltrion | Phase 1 | Completed | |
| CT-L01 12.5/500 mg + Alogliptin Benzoate 12.5 mg + Metformin HCl XR 500 mg | Celltrion | Phase 1 | Completed | |
| L04RD1 + L04TD2 + L04TD2 + L04RD1 | Celltrion | Phase 1 | Completed | |
| CT-P39 + EU-approved Xolair + CT-P39 + EU-approved Xolair + US-licensed Xolair | Celltrion | Phase 1 | Completed | |
| CT-P17 + CT-P17 | Celltrion | Phase 1 | Completed | |
| CSL112 + Placebo | CSL | Phase 1 | Completed | |
| UT-15C | United Therapeutics | Phase 1 | Completed | |
| TP-05 (lotilaner oral), fasted group + TP-05 (lotilaner oral), high-fat group + TP-05 (lotilaner oral), low-fat group | Tarsus Pharmaceuticals | Phase 1 | Completed | |
| TP-03 (Lotilaner Ophthalmic Solution), 0.25% | Tarsus Pharmaceuticals | Phase 1 | Completed | |
| TP-05 (lotilaner oral capsules) + Placebo | Tarsus Pharmaceuticals | Phase 1 | Completed | |
| MBX 2109 (Part A) + MBX 2109 (Part B) + Placebo | MBX Biosciences | Phase 1 | Completed | |
| Dabigatran etexilate + Rosuvastatin + Daridorexant | Idorsia | Phase 1 | Completed | |
| Daridorexant + Famotidine + Efavirenz | Idorsia | Phase 1 | Completed | |
| Open-label TRV734 125 mg + TRV734 blinded + Oxycodone IR 10 mg + Placebo | Trevena | Phase 1 | Completed | |
| TRV130 + Moxifloxacin + Placebo | Trevena | Phase 1 | Completed | |
| Radiolabeled TRV130 | Trevena | Phase 1 | Completed | |
| TRV130A + Dextrose in Water | Trevena | Phase 1 | Completed | |
| TRV734 | Trevena | Phase 1 | Completed | |
| Nalmefene | Tharimmune | Phase 1 | Completed | |
| THB335 single dose + Single dose placebo + THB335 fasted/fed + Placebo fasted/fed + THB335 multiple dose + Multiple dose placebo | Third Harmonic Bio | Phase 1 | Completed | |
| AL002 | Alector | Phase 1 | Completed | |
| AL001 | Alector | Phase 1 | Completed | |
| AL101 | Alector | Phase 1 | Completed | |
| AL003 | Alector | Phase 1 | Completed | |
| SYNB8802 + Placebo | Synlogic | Phase 1 | Completed | |
| CDX-6114 + Placebo | Codexis | Phase 1 | Completed | |
| CDX-6114 + Placebo | Codexis | Phase 1 | Completed | |
| SYNB1934 + SYNB1618 | Synlogic | Phase 1 | Completed | |
| Propranolol + Pseudoephedrine | Eli Lilly | Pre-clinical | Completed | |