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Don Bergstrom, M.D., Ph.D.

President of Research and Development

Relay Therapeutics

Therapeutic Areas

Relay Therapeutics Pipeline

DrugIndicationPhase
RLY-4008 (lirafugratinib)FGFR2-altered solid tumors (e.g., cholangiocarcinoma)Phase 1/2
RLY-2608PI3Kα-mutant solid tumors (e.g., breast cancer)Phase 1
GDC-1971 (formerly RLY-1971)SHP2 inhibition in solid tumorsPhase 1
RLY-2139CDK2 inhibition in solid tumorsPreclinical
Undisclosed ProgramMutant RAS (KRAS G12C & beyond)Discovery